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  • 產品名稱:AZD-0156

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AZD-0156
詳情介紹:
Purpose A potent Ataxia Telangiectasia Mutated (ATM) kinase inhibitor
Characteristics AZD-0156 is an orally bioavailable Ataxia Telangiectasia Mutated (ATM) kinase inhibitor, with potential chemo-/radio-sensitizing and antineoplastic activities. AZD-0156 targets and binds to ATM, thereby inhibiting the kinase activity of ATM and ATM-mediated signaling.
Purity ≥ 98?% by HPLC
Chemical Name 8-[6-[3-(dimethylamino)propoxy]-3-pyridyl]-3-methyl-1-tetrahydropyran-4-yl-imidazo[4,5-c]quinolin-2-one
Formula C??H??N?O?
Permeability Cell-permeable
Solubility DMSO
Molecular Weight 461.57 g/mol
CAS-No 1821428-35-6
Restrictions For Research Use only
Format Solid
Handling Advice Protect from air and light
Storage -20 °C
Expiry Date 36 months